Book Chapters | wdlubellgroup

• Book Chapters

9. Chingle, R.; Lubell, W.D. “(6-Chloro-1-hydroxybenzotriazol-l-y- N-oxy-tris(pyrrolidino)phosphonium Hexafluorophosphate (PyClock)” Encyclopedia of Reagents for Organic

Synthesis (e-EROS), 2017. A. B. Charette, J. W. Bode, T. Rovis, P. L. Fuchs (Eds); John Wiley & Sons Ltd.: Chichester, in press.

8. Chingle, R.; Lubell, W.D. “O-(6-Chlorobenzotriazol-1-yl)-N,N, N′,N′-tetramethyluronium Hexafluorophosphate (HCTU)” Encyclopedia of Reagents for Organic Synthesis (e-

EROS), 2017. A. B. Charette, J. W. Bode, T. Rovis, P. L. Fuchs (Eds); John Wiley & Sons Ltd.: Chichester, in press.

7. St-Cyr, D.J.; García-Ramos, Y.; Doan, N.-D.; Lubell, W.D. “Aminolactam, N-Aminoimidazolone, and N-Aminoimdazolidinone Peptide Mimics” in Peptidomimetics I, Series:

Topics in Heterocyclic Chemistry, W. Lubell (Ed.) Vol. 48, 2017, 125-175. ISBN 978-3-319-49119-6

6. Bourguet CB, Lubell WD. “Synthesis and alkylation of Aza-Gly-Pro building blocks of peptidomimetic libraries for developing prostaglandin F2α receptor modulators as

therapeutics to inhibit preterm labor.” Methods Mol. Biol. 2015; 1248: 81-91. doi: 10.1007/978-1-4939-2020-4_6.

5. Proulx, C.; Lubell, W. D. “O-(3,4-Dihydro-4-oxo-1,2,3-benzotriazin-3-yl)-N,N,N’,N’-tetramethyl-uronium tetrafluoroborate” Encyclopedia of Reagents for Organic Synthesis, 2012.

A. B. Charette, D. Crich, P. L. Fuchs, G. A. Molander (Eds); John Wiley & Sons Ltd.: Chichester, 2nd Ed.; (I.D.: RN01543), 2013.

4. Proulx, C.; Lubell, W. D. “O-(6-Chloro-1H-benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium tetra-fluoroborate” Encyclopedia of Reagents for Organic Synthesis, 2012. A. B.

Charette, D. Crich, P. L. Fuchs, G. A. Molander (Eds); John Wiley & Sons Ltd.: Chichester, 2nd Ed.; (I.D.: RN01544), 2013.

3. Lubell, W. D.; St-Cyr, D. J.; Dufour-Gallant, J.; Hopewell, R.; Boutard, N.; Kassem, T.; Dörr, A.; Zelli, R., “1H-Pyrroles” In Science of Synthesis Knowledge Updates, Fuerstner,

A., Ed.; Thieme: Stuttgart, (2013); Vol. 2013/1, Section 9.13.5, p 157-408.

2. K. Beauregard, F. Polyak, W. D. Lubell (2012) Peptides and Chirality Effects on the Conformation and the Synthesis of Medicinally Relevant Peptides. In: Carreira E.M. and

Yamamoto H. (eds.) Comprehensive Chirality, Volume 1, pp. 86-104. Amsterdam: Elsevier.

1. W. D. Lubell, J. W. Blankenship, G. Fridkin, and R. Kaul (2005) “Peptides.” Science of Synthesis 21.11, Chemistry of Amides. Thieme, Stuttgart, 713-809.

• Editorials and Book Reviews

4. Papini, A.M.; Lavielle, S.; Lubell, W.D. “Peptides in Paris” Biopolymers. 2015, 104, v-vii. doi: 10.1002/bip.22738.

3. Lubell, W. D. “Peptide Chemistry” editorial for virtual issue of Org. Lett., J. Org. Chem. And J. Am. Chem. Soc. 2012 online Sept. 7.

2. Lubell WD. Editorial “Thoughts on Meldal and Hirschmann.” Biopolymers. 2010; 94(2): iii-v. doi: 10.1002/bip.21373.

1. lubell, w. Book Review of "Solid-Phase Organic Synthesis." Edited by Kevin Burgess, for J. Am. Chem. Soc. 2001, 123, 6744.

• Books

3. W. Lubell (Ed.) Peptidomimetics I Series: Topics in Heterocyclic Chemistry, Vol. 48, 2017, ISBN 978-3-319-49119-6

2. W. Lubell (Ed.) Peptidomimetics II Series: Topics in Heterocyclic Chemistry, Vol. 49, 2017, ISBN 978-3-319-49124-0

1. “Advances in Experimental Medicine and Biology” volume 611, “Peptides for Youth, Proceedings of the 20th American Peptide Society Meeting”, S. E. Del Valle, E. Escher, W.

D. Lubell, Editors, 2009, Springer Science, (ISBN: 978-0-387-73656-3).

• Refereed Proceedings of American, Japanese and European Peptide Symposia

72. Poupart, J.; Lubell, W.D. “4,5-Disubstituted N-aminoimdazol-2-One Mimics of Peptide Turn Backbone and Side Chain Conformation” Proceedings of the 24th American Peptide

Symposium, Ved Srivastava, Andrei Yudin, and Michal Lebl (Editors) American Peptide Society, 2015, 272-273.

71. Traore, M.; Lubell W.D. “Solid-Phase Synthesis of Aza-Lysine Peptide Analogue of Trypsin Substrate” Proceedings of the 24th American Peptide Symposium, Ved Srivastava,

Andrei Yudin, and Michal Lebl (Editors) American Peptide Society, 2015, 187-188.

70. Mohammadpour, F,; Chemtob, S.; Hou, X.; Lubell W.D. “Synthesis and Evaluation of Azapeptide Prostaglandin F2α Receptor Modulators in Pursuit of Inhibitors of Preterm

Labor” Proceedings of the 24th American Peptide Symposium, Ved Srivastava, Andrei Yudin, and Michal Lebl (Editors) American Peptide Society, 2015, 187-188.

69. Merlino, F.; Yousif, A. M.; Di Maro, S.; Turcotte, S.; Dufour-Gallant, J.; Chatenet, D.; Santicioli, P.; Novellino, E.; Grieco, P.; Lubell, W.D. “Synthesis of N-Methyl and Azasulfuryl

Urotensin-II(4-11) Derivatives” Proceedings of the 24th American Peptide Symposium, Ved Srivastava, Andrei Yudin, and Michal Lebl (Editors) American Peptide Society,

2015, 184-186.

68. Chingle, R.; Lubell, W.D. “Peptide coupling challenges in azopeptide route to aza-pipecolyl Smac mimetic” Proceedings of the 24th American Peptide Symposium, Ved

Srivastava, Andrei Yudin, and Michal Lebl (Editors) American Peptide Society, 2015, 172-173.

67. Poupart, J.; Lubell, W.D. "Mitsunobu Reaction on Solid Support for Peptide N-terminal Farnesylation" Proceedings of the 24th American Peptide Symposium, Ved Srivastava,

Andrei Yudin, and Michal Lebl (Editors) American Peptide Society, 2015, 94-95.

66. Turcotte, S.; Lubell, W.D. "Solid-Phase Synthesis of Azasulfurylphenylalanine4-GHRP-6" Proceedings of the 24th American Peptide Symposium, Ved Srivastava, Andrei Yudin,

and Michal Lebl (Editors) American Peptide Society, 2015, 40-42.

65. Doan, N.-D.; Lubell, W.D. “Solid-Phase Synthesis of Z-alkene Aza-Lysine Peptidomimetics” Proceedings of the 33rd European Peptide Symposium, Emilia Naydenova, Tamara

Pajpanova (Editors) European Peptide Society, 2014, 4-5.

64. Yésica García-Ramos, William D. Lubell “Synthesis of Azapeptide Ligands of the CD36 Receptor Towards Potential Treatments of Age-Related Macular Degeneration ” In

Peptides 2013 (Proceedings of the 23rd American Peptide Symposium 2013), M. Lebel Editor, 2013, 188-189.

63. Yésica García-Ramos, Caroline Proulx, William D. Lubell “Analysis of N-Amino-Imidazolidin-2-one Turn Mimic Geometry” In Peptides 2013 (Proceedings of the 23rd American

Peptide Symposium 2013), M. Lebel Editor, 2013, 190-191.

62. Caroline Proulx, Samir H. Bouayad-Gervais, Yésica García-Ramos, William D. Lubell "N-Amino-imidazolin-2-one turn mimics" Proceedings of the 32nd Europ. Peptide Symp.

(2012) George Kokotos, Violetta Constantinou-Kokotou, John Matsoukas (Eds) European Peptide Society, 2012, pp. 18-19.

61. Stéphane Turcotte, Thierry Havard, William D. Lubell "Mild chemoselective alkylation of aza-sulfurylglycinyl peptides" Proceedings of the 32nd Europ. Peptide Symp. (2012)

George Kokotos, Violetta Constantinou-Kokotou, John Matsoukas (Editors) European Peptide Society, 2012, pp. 140-141.

60. Yésica García-Ramos, Caroline Proulx, Christophe Camy, William D. Lubell "Synthesis and purification of enantiomerically pure N-aminoimidazolin- 2-one dipeptide"

Proceedings of the 32nd Europ. Peptide Symp. (2012) George Kokotos, Violetta Constantinou-Kokotou, John Matsoukas (Editors) European Peptide Society, 2012, pp. 366-

367.

59. Bourguet, C., B.; Lubell, W. D. “On the Nature of Azabicyclo[X.Y.0]alkanone and Aza-dipeptide Mimicry of Turn Conformations” In Peptides 2011 (Proceedings of the 22nd

American Peptide Symposium 2011), M. Lebel Editor, 2011, 82-83. (NSERC, FQRNT, CIHR)

58. Sabatino, D.; Lubell, W. D. “Submonomer Solid-Phase Synthesis of Aza-Glu Peptides” In Peptides 2011 (Proceedings of the 22nd American Peptide Symposium 2011), M.

Lebel Editor, 2011, 78-79.

57. Proulx, C.; Lubell, W. D. “Synthesis of [Azaphenylglycine4]- and [Aza-1-phenyl-2,3-triazole-3-alanine4]Growth Hormone Releasing Peptide-6 and comparison of their

conformations with [AzaPhe4]GHRP-6” In Peptides 2011 (Proceedings of the 22nd American Peptide Symposium 2011), M. Lebel Editor, 2011, 80-81. (NSERC, FQRNT)

56. Ronga, L.; Beauregard, K.; Jamieson, A. G.; St-Cyr, D.; Quiniou, C.; Chemtob, S.; Lubell, W. D. “Structure-activity relationship study of an interleukin-1 receptor negative

modulator by α-amino γ-lactam scanning” In Peptides 2010 (Proceedings of the 31st European Peptide Symposium 2010), M. Lebl, M. Meldal, K. J. Jensen, T. Hoeg-Jensen

Editors, 2010, 256-257. (NSERC, CIHR)

55. Proulx, C., Sabatino, D., Pohankova, P., Ong, H., Lubell, W.D. “Synthesis, conformational analysis, and biological activity of [aza-3-indoylgly4] GHRP-6 as an aza-tryptophan

analog of Growth Hormone Releasing Peptide-6” In Peptides 2010 (Proceedings of the 31st European Peptide Symposium 2010), M. Lebl, M. Meldal, K. J. Jensen, T. Hoeg-

Jensen Editors, 2010, 458-459.

54. Boutard, N.; Dufour-Gallant, J.; Lubell, W.D. “Rapid Synthesis of Pyrrolo[3, 2-e][1, 4]diazepin-2-one γ-Turn Mimics on TAP Soluble Support” In Peptides 2010 (Proceedings of

the 31st European Peptide Symposium 2010), M. Lebl, M. Meldal, K. J. Jensen, T. Hoeg-Jensen Editors, 2010, 268-269.

53. Ronga, L.; Lubell, W. D. “Solid-phase synthesis and CD spectral analysis of IL1R-Allosteric Modulator 101.10 Bearing Multiple Agl-residues” In Peptides 2009 (Proceedings of

the 21st American Peptide Symposium 2009), M. Lebel Editor, 2009, 86-87. (NSERC, CIHR)

52. Boutard, N.; Jamieson, A. G.; Lubell, W. D. “Solid-phase synthesis and CD spectroscopic conformational analysis of alpha- and beta-amino- gamma-lactam (Agl and Bgl)

analogs of growth hormone releasing peptide GHRP-6” In Peptides 2009 (Proceedings of the 21st American Peptide Symposium 2009), M. Lebel Editor, 2009, 78-79. (NSERC,

FQRNT, CIHR)

51. Bourguet, C., B.; Lubell, W. D. “Synthesis of radio-labelled peptide mimic for examining affinity and activity at the prostaglandin F2a receptor” In Peptides 2009 (Proceedings of

the 21st American Peptide Symposium 2009), M. Lebel Editor, 2009, 76-77. (NSERC, FQRNT, CIHR)

50. Sabatino, D.; Lubell, W. D. “Submonomer solid-phase aza-peptide synthesis and circular dichroism spectroscopic analysis of [aza-Phe4]-GHRP-6” In Peptides 2009

(Proceedings of the 21st American Peptide Symposium 2009), M. Lebel Editor, 2009, 58-59. (NSERC, FQRNT)

49. Proulx, C.; Lubell, W. D. “Solid-phase synthesis of aza-Pro analogs of GHRP-6” In Peptides 2009 (Proceedings of the 21st American Peptide Symposium 2009), M. Lebel

Editor, 2009, 56-57.

48. Deaudelin, P.; Iden, H.; Lubell, W.D. “Solution- and solid-phase chemistry for the synthesis of diazepinones and structural proof for their mimicry of g-turn conformations” In

Peptides 2008 (Proceedings of the 30th European Peptide Symposium 2008), 198-199.

47. Iden, H. S.; Lubell. W. D. “Solid-Phase Synthesis of a 1,3,5-Trisubstituted 1,4-Diazepin-2-one Peptide Mimic” In Peptides 2007 (Proceedings of the 21st American Peptide

Symposium 2007) E. Escher, W. D. Lubell, S. E. Del Valle, Eds, 2009, 213-214.

46. Lama, T,; Singer, R. D.; Lubell; W. D. “Peptides of Life Teaching Peptide Science and Art in Elementary School” In Peptides 2007 (Proceedings of the 21st American Peptide

Symposium 2007) E. Escher, W. D. Lubell, S. E. Del Valle, Eds, 2009, lxxi - lxxiii.

45. Bourguet, C. B.; Dörr, A.; Godina, T.; Proulx, C.; Fridkin, G.; Jamieson, A., Sabatino, D., Kassem, T.; Boutard, N.; Aresenault, J.; Ronga, L.; Brouillette, Y.; Bednarek, M.; Tolle,

J. C.; Lubell, W.D. “Portraits of the Pioneers of the American Peptide Society” In Peptides 2007 (Proceedings of the 21st American Peptide Symposium 2007) E. Escher, W. D.

Lubell, S. E. Del Valle, Editors, 2009, xlix - lxix.

44. Proulx, C.; Sabatino, D.; Godina, T.; Lubell, W. D. “’Experiment’, a pictorial retrospective from the first peptide bond to the 20th American Peptide Society Meeting” In Peptides

2007 (Proceedings of the 21st American Peptide Symposium 2007) E. Escher, W. D. Lubell, S. E. Del Valle, Editors, 2009, xxxiii - xlviii.

43. Kassem, T.; Zhu, X.X.; Lubell. W. D. Poly (ethylene glycol) Supported Hydroxyproline: Application in the Asymmetric Aldol Reaction” In Peptides 2007 (Proceedings of the 21st

American Peptide Symposium 2007) S. E. Del Valle, E. Escher, W. D. Lubell, Editors, 2009, 223-4.

42. Genest, N.; Lama, T.; Seaman, S. E.; Lubell, W. D. “Towards an Efficient Synthesis of Hydroxyethylene Dipeptide Isostere of Phe-Aib” In Peptides 2007 (Proceedings of the

21st American Peptide Symposium 2007) S. E. Del Valle, E. Escher, W. D. Lubell, Eds, 2009, 221-222.

41. Lama, T.; Fridkin, G.; Lubell, W. D. “Poly-(Proy[CH(OAc)CH2]Aib)3 a Protected Trimer of Pro-Aib Hydroxyethylene Isosteres” In Peptides 2007 (Proceedings of the 21st

American Peptide Symposium 2007) S. E. Del Valle, E. Escher, W. D. Lubell, Ed., 2009, 171-2

40. Dörr, A.; Lubell, W.D. “Synthesis and Peptide Coupling of Protected Pyrrolylalanine” In Peptides 2007, S. E. Del Valle, E. Escher, W. D. Lubell, Editors, 2009 (Proceedings of

the 21st American Peptide Symposium 2007) 217-218.

39. Bourguet, C.B. ; Hou, X.; Chemtob, S.; Lubell, W. D. “Exploring the relationship between turn geometry and allosteric antagonism of peptide mimic ligands for the

prostaglandin F2alpha receptor” In Peptides 2007 (Proceedings of the 21st American Peptide Symposium 2007) S. E. Del Valle, E. Escher, W. D. Lubell, Editors, 2009, 271-2.

38. Ben tahar, W. B.; Keillor, J. W.; Lubell. W. D. “Microwave synthesis of fluorescent tags” In Peptides 2007 (Proceedings of the 21st American Peptide Symposium 2007) S. E.

Del Valle, E. Escher, W. D. Lubell, Editors, 2009, 225-6.

37. Deaudelin, P.; Lubell. W. D. “Synthesis of pyrrolo[3,2-e][1,4]diazepinon-2-ones as potential g-turn mimics” In Peptides 2007 (Proceedings of the 21st American Peptide

Symposium 2007) E. Escher, W. D. Lubell, S. E. Del Valle, Editors, 2009, 183-184.

36. Iden, H. S.; Lubell. W. D. “1,3,5-Trisubstituted 1,4-Diazepin-2-one Synthesis” Proceedings of 43JPS/PEM4 2006, Hitoshi Ishida and Hisakazu Mihara (Eds), Japanese Peptide

Society, 2006, 24-25.

35. Dorr, A., Lubell. W. D. “The Influence of p-Deficient Phenylalanine Derivatives on Prolyl Amide Isomer Population” Proceedings of 43JPS/PEM4 2006, Hitoshi Ishida and

Hisakazu Mihara (Editors), Japanese Peptide Society, 2006, 68-69.

34. Lama, T.; Seaman, S. E.; Genest, N.; Lubell, W. D. «Synthesis and Conformational Analysis of a Pro-Aib Hydroxyethylene Dipeptide Isostere« In Peptides 2006 (Proceedings

of the 29th European Peptide Symposium 2006), K. Rolka, P. Rekowski, J. Silberring Editors, 2006, 432-433.

33. Bourguet, C.B.; Hou, X.; Chemtob, S.; Lubell, W. D. «Influence of Peptide Mimic Turn Stereochemistry on Allosteric Antagonism at the Prostaglandin F2a Receptor” In Peptides

2006 (Proceedings of the 29th European Peptide Symposium 2006), K. Rolka, P. Rekowski, J. Silberring Editors, 2006, 436-437.

32. Bodas, M.; Lev-Goldman, V.; Ben-Aroya, N. Koch, Y.; Fridkin, M.; Lubell, W. D. « Freidinger Lactam Scan of LHRH using Fmoc-Protected Cyclic Sulfamidate Methyl Ester ” In

Peptides 2006 (Proceedings of the 29th European Peptide Symposium 2006), K. Rolka, P. Rekowski, J. Silberring Editors, 2006, 528-529.

31. Boeglin, D., R.; Bodas, M. S.; Galaud, F.; Lubell, W. D. " Positional Scanning for Peptide Secondary Structure by Solid Phase Synthesis with Aza-amino acids and Freidinger

lactams" In Peptides 2005 S. E. Blondelle (Editor), American Peptide Society, 2005, 50-51.

30. Boeglin, D., R.; Rao, M. H.V. R.; Demers, J.-P.; Lubell, W. D. "Aza-peptides with multiple aza-amino acids, synthesis and … analysis of Glu-azaAla-Ala-azaAla-Leu-azaAla-

Lys-azaAla-NH2" In Peptides 2005 S. E. Blondelle (Editor), Am. Peptide Society, 2005, 184-5.

29. Galaud, F.; Demers, A.; Ong, H.; Lubell, W. D. "Synthesis and Incorporation of Freidinger Lactam Analogs in GHRP-6 In Peptides 2005 S. E. Blondelle (Ed.), Am. Peptide

Society, 2005, 188-9.

28. Rombouts, F.; Lubell, W. D. "Synthesis of polyfunctionalized pyrrolo[3,2-d] pyrimidines..." In Peptides 2004 (Proceedings of the 28th European Peptide Symp.), J. Slaninova,

Ed., 2004, 577-578.

27. Blankenship, J.; Bélec, L.; Lubell, W. D. "Conformational Analysis of the Oxytocin Antagonists..." In Peptides 2004 (Proceedings 28th Eur. Peptide Symp.), J. Slaninova, Ed.

2004, 85-88.

26. Blankenship, J.; Lubell, W. D. "...Pyrrolo[3,2-d]pyrimidines for application as beta-sheet mimics." In Peptides 2004 (Proceedings of the 28th European Peptide Symposium), J.

Slaninova, Editor, 2004, 746-747.

25. Melendez, R. E.; Lubell, W. D. "Synthesis of azapeptides using N-Boc-aza1-dipeptide building blocks." In Peptides 2003 M. Chorev and T. Sawyer, Editors, 2004, 37-38.

24. Galaud, F.; Laborde, P.; Lubell, W. D. "Peptide Mimic Synthesis with Cyclic Sulfamidates" In Peptides 2003 M. Chorev and T. Sawyer, Editors, 2004, 188-189.

23. Dettwiler, J.E.; Bélec, L.; Lubell, W. D. "...Study of an aureobasidin peptide antibiotic: synthesis of Boc-N-methylhydroxyvaline" In Peptides 2003 M. Chorev and T. Sawyer,

Eds, 2004, 179-180.

22. Jeannotte, G., Hansford, K.A.;Marcotte, Frederik, F.-A.; Rombouts, F.; Zanzarova, V.; Lubell, W. D. "Aminopyrrole Carboxylates...." In Peptides 2003 M. Chorev & T. Sawyer,

Eds, 2004, 176-178.

21. Jeannotte, G.; Lubell, W. D. "Synthesis and Use of Pyrrol-Prolines for Peptide Mimicry." In Peptides 2002 (Proceedings of the 27th European Peptide Symposium), E.

Benedetti, Editor, 2002, 206-207

20. Dietrich, E.; Lubell, W. D. "Il mondo é bello perché é varioî, expanding azabicycloalkanone amino acid diversity. Efficient Synthesis of pyrrolizidinone amino acid." In Peptides

2002 (Proceedings of the 27th European Peptide Symposium), E. Benedetti, Editor, 2002, 202-203.

19. Melendez, R. E.; Lubell, W. D. "Novel Approach for Enantiopure Azapeptide Synthesis..." In Peptides 2002 (Proceedings of the 27th European Peptide Symposium), E.

Benedetti, Editor, 2002, 204-205.

18. Cluzeau, J.; Lubell, W. D. "Mimicry of ... Peptide Turns: Synthesis of Novel 4-Substituted Indolizidin-9-one Amino Acids." In Peptides, M. Lebel & R. Houghten, Eds, 2001, 597-

598.

17. w. d. "Employing the steric interactions of 5-tert-butylproline to control peptide folding and biology" In Peptides, M. Lebel and R. Houghten, Eds, 2001, 599-601.halab, L.; Bélec,

l.; lubell

16. dairi, k.; keillor, j.w.; lubell, w. d. "Solid-Phase Synthesis of Aspartic Protease" In Peptides 2000, J. Martinez & J.-A. Fehrentz, Eds. EDK, Paris, 2001, 803-804.

15. halab, L.; lubell, w. d. "Stabilization of Type VI b-Turns in Tetrapeptides" In Peptides 2000 J. Martinez & J.-A. Fehrentz, Eds. EDK, Paris, 2001, 815-816.

14. bélec, l.; slaninova, j.; lubell, w.d. "Steric Interactions of Penicilamine6-5-tert-Butylproline7-Oxytocin Analogs..." In Peptides 2000, J. Martinez & J.-A. Fehrentz, Eds. EDK, Paris,

2001, 587-8.

13. Lubell, W. D.; miranda, l.; meldal, m. HYDRA: A Novel Hydroxy and Amine Resin"In Peptides 2000 , J. Martinez & J.-A. Fehrentz, Eds. EDK, Paris, 2001, 981-982.groth, t.;

grøtli, m.; lubell

12. polyak, f.; lubell, w. d. “Mimicry of Peptide Back-bone and Side-Chain Functions: Syntheses of 5- and 7-Hydroxymethyl Indolizidinone Amino Acids and Indolizidinone Amino

Dicarboxylate, Constrained Ser-Pro and Glu-Pro Surrogates” In Peptides, G. Fields & G. Barany, Eds, 2000, 150-1.

11. bélec, l.; slaninova, j.; lubell, w. d. "Studying the influence of prolyl amide geometry on bioactivity with 5-t-BuPro oxytocin analogs." In Peptidess, G. Fields & G. Barany, Eds,

2000, 630-1.

10. Lubell, w. d. "The effects of stereochemistry and sequence on 5-10 halab, L.; lubelltert-butylproline type VI b-turn mimics." In Peptides: Chem., Structure and Biology, G.

Fields & G. Barany, Eds; 2000, 305-6.

9. gosselin, f.; swarbrick, m. e.; lubell, w. d. "Synthesis of e-Alkylpipecolates as Conformationally Rigid Proline Surrogates" Peptides 1998 (Proceedings of the 25th Europ. Peptide

Symp.), S. Bajusz & F. Hudecz, Eds; Akadémia Kiadó, Budapest, Hungary, 1999, 678-679.

8. halab, L.; lubell, w. d. "Steric Effects of 5-tert-Butylproline in Dipeptide Mimics of Type VI b-Turns." In Peptides 1998 (Proceedings of the 25th European Peptide Symposium), S.

Bajusz and F. Hudecz, Editors; Akadémia Kiadó, Budapest, Hungary, 1999, 356-357.

7. polyak, f.; lubell, w. d. "Synthesis and Incorporation of 7-Benzyl Indolizidinone Amino Acid into Leucine Enkephalin." In Peptides 1998 (Proceedings of the 25th European

Peptide Symposium), S. Bajusz and F. Hudecz, Editors; Akadémia Kiadó, Budapest, Hungary, 1999, 688-689.

6. gosselin, f.; lubell, w. d. "Indolizidin-9-one Amino Acid, A New Rigid Dipeptide Turn Mimic." In Peptides 1998 (Proceedings of the 25th European Peptide Symposium), S. Bajusz

and F. Hudecz, Editors; Akadémia Kiadó, Budapest, Hungary, 1999, 660-661.

5. beausoleil, e.; lubell, w.d. "Steric Effects of 5-tert-Butylproline on the Conformation of Polyproline." In Peptides: Chem., Structure and Biology, James P. Tam & P.T.P.

Kaumaya, Eds; ESCOM, Leiden, The Netherlands, 1998, 150-151.

4. michnick, S.; lubell, w.d. "Steric Effects of Alkylprolines on the Conformation of N-(Acetyl)Proline N'-Methylamides". In Peptides 1996 (Proceedings of the 24th Europ. Peptide

Symp.), R. Ramage & R. Epton, Eds; ESCOM, Leiden, The Netherlands, 1997, pp 241-242.beausoleil, e.; sharma

3. lombart, h.-g.; lubell, w. d. "Use Of Azabicycloalkane Amino Acids To Stabilize b-Turn Conformations In Model Peptides And Gramicidin S". In Peptides: Chemistry, Structure

and Biology, P.T.P. Kaumaya and R.S. Hodges , Editors; ESCOM Sci. Pub. B.V.: Leiden, The Netherlands, 1996, 695-696.

2. lombart, h.-g.; lubell, w. d. "A Claisen Condensation Approach To Prepare Azabicycloalkane Amino Acid b-Turn Mimetics". In Peptides 1994 (Proceedings of the 23rd European

Peptide Symposium), H. L. S. Maia, Ed.; ESCOM, Leiden, Netherlands, 1995, 696-7.

1. beausoleilatfani, m.; lubell, w. d. "Synthesis Of 5-Alkylprolines And Their Use In The Design Of X-Proline Cis-Amide Surrogates". In Peptides: Chemistry, Structure and Biology,

R.S. Hodges and J.A. Smith, Editors; ESCOM Science Publishers B.V.: Leiden, The Netherlands, 1994, 307-309., h. h.; ibrahim